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Search Results for " glucocorticoid receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
T37908 Glucocorticoid receptor agonist-1 Glucocorticoid Receptor
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].
T11417 Glucocorticoid receptor agonist Others
Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.
T67742 EX-A5386 Glucocorticoid receptor modulator-1 Glucocorticoid Receptor
EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.
T63551 Glucocorticoid receptor-IN-1
Glucocorticoid receptor-IN-1 is a selective regulator of the glucocorticoid receptor (GR) and exhibits anti-inflammatory activity. glucocorticoid receptor-IN-1 has good transcriptional repression, acting on hMMP1 ( IC50:...
T63539 Glucocorticoid receptor-IN-2
Glucocorticoid receptor-IN-2 is a selective regulator of the glucocorticoid receptor (GR) and exhibits anti-inflammatory activity. IC50: 0.171 nM) and also has some transcriptional activating effect on MMTV (EC50: 0.94 n...
T72102 Glucocorticoid receptor modulator 1
Glucocorticoid receptor modulator 1 is a potent, orally active, non-steroidal selective glucocorticoid receptor modulator, exhibiting IC50 values of 9 nM and 130 nM against NF-κB and AP-1, respectively. It effectively re...
T74697 Glucocorticoid receptor agonist-2
Glucocorticoid receptor agonist-2 (compound 21), a glucocorticoid receptor agonist exhibiting an IC50 value of 6.6 nM, serves as an active reference for ABBV-3373 [1]. This compound is instrumental in the synthesis of an...
T15451 GW-870086 Glucocorticoid Receptor
GW-870086 is an effective anti-inflammatory agent. GW-870086 also plays a role in a glucocorticoid receptor agonist (pIC50: 10.1 in A549 cells expressing NF-κB).
T14377 AZD5423 Glucocorticoid Receptor
AZD5423 is an inhaled, potent, selective, and non-steroidal modulator of glucocorticoid receptor (GR) and it effectively reduces allergen-induced responses in subjects with mild allergic asthma.
T8777 Beclometasone BecloMethasone Glucocorticoid Receptor
Beclometasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma.
T14981 Clobetasone butyrate Glucocorticoid Receptor
Clobetasone butyrate, a synthetic glucocorticoid with topical anti-inflammatory activity, is effective in treating corticosteroid-responsive dermatoses, such as atopic dermatitis and psoriasis, especially within skin tis...
T1560 Prednisolone Predonine,Hydroretrocortine,Metacortandralone Glucocorticoid Receptor , Endogenous Metabolite
Prednisolone (Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.
T1614 Hydrocortisone Cortisol Glucocorticoid Receptor , Endogenous Metabolite
Hydrocortisone (Cortisol) is a glucocorticoid hormone secreted by the adrenocortex. Hydrocortisone agonizes the glucocorticoid receptor, which promotes proteolytic metabolism, gluconeogenesis, capillary wall stabilizatio...
T17217 Vamorolone VBP15 Glucocorticoid Receptor , NF-κB
Vamorolone (VBP15) is an orally active dissociative steroidal anti-inflammatory drug and membrane-stabilizer. Vamorolone improves muscular dystrophy without side effects. Vamorolone displays effective NF-κB inhibition an...
T1168 Desonide Tridesilon,Locapred,Prednacinolone Glucocorticoid Receptor
Desonide (Prednacinolone) is a synthetic glucocorticosteroid for topical use, with anti-inflammatory activity. Desonide binds to glucocorticoid receptors in the cytoplasm, and the ligand-receptor complex is translocated ...
T0798 Triamcinolone Fluoxyprednisolone,Aristocort,Rodinolone Glucocorticoid Receptor , COX
Triamcinolone (Aristocort) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties. Upon cell entry, triamcinolone binds to and activates the glucocorticoid receptor, which leads to transloca...
T0820 Triamcinolone acetonide Aristogel,Azmacort,Aristoderm Glucocorticoid Receptor
Triamcinolone acetonide (Azmacort) is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as a Corticosteroid Hormone Receptor Agonist. It is an anti-inflammatory glucocorticoid used topically in the ...
T74116 Glucocorticoid receptor agonist-1 Ala-Ala-Mal
Glucocorticoid receptor agonist-1 Ala-Ala-Mal (compound 88), a glucocorticosteroid and glucocorticoid receptor agonist, can be conjugated with Adalimumab to formulate an ADC [1].
T77869 Glucocorticoid receptor agonist-2 Ala-Ala-Mal
Glucocorticoid receptor agonist-2 Ala-Ala-Mal (compound 79) serves as a precursor for synthesizing anti-inflammatory antibody-drug conjugate (ADC) molecules and acts as an active reference for ABBV-3373 [1].
T6502 Fluocinonide Lidex,Metosyn,Topsyn Glucocorticoid Receptor
Fluocinonide (Topsyn) (Vanos) is an effective glucocorticoid steroid, utilized in the treatment as the skin disorders anti-inflammatory agent.

Compounds

Glucocorticoid receptor agonist-1
T37908
Synonym:
Target: Glucocorticoid Receptor
Glucocorticoid receptor agonist
T11417
Synonym:
Target: Others
EX-A5386
T67742
Synonym: Glucocorticoid receptor modulator-1
Target: Glucocorticoid Receptor
Glucocorticoid receptor-IN-1
T63551
Synonym:
Target:
Glucocorticoid receptor-IN-2
T63539
Synonym:
Target:
Glucocorticoid receptor modulator 1
T72102
Synonym:
Target:
Glucocorticoid receptor agonist-2
T74697
Synonym:
Target:
GW-870086
T15451
Synonym:
Target: Glucocorticoid Receptor
AZD5423
T14377
Synonym:
Target: Glucocorticoid Receptor
Beclometasone
T8777
Synonym: BecloMethasone
Target: Glucocorticoid Receptor
Clobetasone butyrate
T14981
Synonym:
Target: Glucocorticoid Receptor
Prednisolone
T1560
Synonym: Predonine,Hydroretrocortine,Metacortandralone
Target: Glucocorticoid Receptor, Endogenous Metabolite
Hydrocortisone
T1614
Synonym: Cortisol
Target: Glucocorticoid Receptor, Endogenous Metabolite
Vamorolone
T17217
Synonym: VBP15
Target: Glucocorticoid Receptor, NF-κB
Desonide
T1168
Synonym: Tridesilon,Locapred,Prednacinolone
Target: Glucocorticoid Receptor
Triamcinolone
T0798
Synonym: Fluoxyprednisolone,Aristocort,Rodinolone
Target: Glucocorticoid Receptor, COX
Triamcinolone acetonide
T0820
Synonym: Aristogel,Azmacort,Aristoderm
Target: Glucocorticoid Receptor
Glucocorticoid receptor agonist-1 Ala-Ala-Mal
T74116
Synonym:
Target:
Glucocorticoid receptor agonist-2 Ala-Ala-Mal
T77869
Synonym:
Target:
Fluocinonide
T6502
Synonym: Lidex,Metosyn,Topsyn
Target: Glucocorticoid Receptor
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TargetMol